Kudzorerazve (LY3437943)ipeptide yekugadzira yechizvarwa chinotevera yakagadzirwa seagonist yekugamuchira katatuinotarisa GLP-1, GIP, uye glucagon receptors. Dhizaini yayo itsva yemamorekuru inoisiyanisa netekinoroji yekare ye single- uye dual-receptor peptide, zvichiita kuti ive imwe yemakemikari akanyanya kudzidzwa muongororo yemazuva ano ye metabolic.
Inopihwa seupfu hwakachena kwazvo hwakasanganiswa ne lyophilized,Kudzorerazveinopa kugadzikana kwakanaka pakubata, kutakurwa, uye kuchengetwa kwenguva refu. Inowanzoshandiswa mukuferefeta kwesainzi kunosanganisira receptor signaling, metabolic regulation, peptide engineering, uye endocrine research.
✔ Kuchena Kwakanyanya (≥98% HPLC)
✔ Upfu hwakacheneswa kusvika kuchena husina kuchena
✔ Kugadzikana Kwakanaka Kwemapurogiramu Ekutsvaga
✔ Tekinoroji yeAgonist yeTriple Receptor
✔ Kudzora Hunhu Hwakasimba uye Kuenderana KwemaBatch
✔ Yakakodzera Kutsvagurudza Kwepamusoro kwePeptide
| Chinhu | Tsanangudzo |
|---|---|
| Zita rechigadzirwa | Kudzorerazve |
| Zita rinoenderana | LY3437943 |
| Fomura yeMolecular | C221H342N46O68* |
| Kurema kweMorekuru | Inenge 4731 Da* |
| Chitarisiko | Upfu hwakachena hwakanyoroveswa |
| Kuchena | ≥98% neHPLC |
| Kuchengetera | -20°C Zvinokurudzirwa |
| Kunyunguduka | Mvura Inonyungudika |
| Kushandiswa | Tsvagiridzo yeLabhoritari Chete |
*Magadzirirwo anogona kusiyana zvichienderana nekugadzirwa kwezvinhu uye mwero wekuongorora.
| Zita rechigadzirwa | Nhamba yeCAS |
|---|---|
| AOD-9604 | 221231-10-3 |
| BPC-157 | 137525-51-0 |
| PT-141 / Bremelanotide Acetate | 189691-06-3 |
| CJC-1295 | 863288-34-0 |
| GHK-Cu | 89030-95-5 |
| GHRP-2 | 158861-67-7 |
| Hexarelin | 140703-51-1 |
| IGF-1 LR3 | 946870-92-4 |
| Ipamorelin | 170851-70-4 |
| KPV / Alpha MSH (11-13) | 67727-97-3 |
| L-Arginine | 74-79-3 |
| MOTS-C | 1627580-64-6 |
| Oxytocin | 50-56-6 |
| PDA | 106-50-3 |
| Selank | 129954-34-3 |
| Semax | 80714-61-0 |
| Sermorelin | 86168-78-7 |
| SS-31 (Lyo) / Elamipretide | 736992-21-5 |
| Chidimbu cheTB500 | 476014-70-7 |
| Tesamorelin | 218949-48-5 |
| Thymogen / Oglufanide | 38101-59-6 |
| Thymosin Alpha-1 / Thymalfasin | 62304-98-7 |
| Thymosin Beta-4 | 77591-33-4 |
| TB500 | 885340-08-9 |
| NVG-291 | 2135482-62-7 |
| CB4211 | 2361287-87-0 |
| DSIP | 62568-57-4 |
| Epitalon | 307297-39-8 |
| Gonadorelin | 33515-09-2 |
| LL-37 | 154947-19-0 |
| Melanotan II | 121062-08-6 |
| MK-0616 | 2249825-14-7 |
| NAD+ | 53-84-9 |
| Pamorelin | 57773-63-1 |
| PTD-DBM | 1241682-11-0 |
| Chidimbu 176-191 | 66004-57-7 |
| VIP | 40077-57-4 |
| PE-22-28 | 1136689-11-0 |
Retatrutide yakagadzirirwa kushanda panguva imwe chete nema metabolic hormone receptors matatu:
Zvinoenderana nekudzora kudya, nzira dzekuburitsa zvinhu mudumbu, uye nzira dzekutumira mashoko dzine chekuita neshuga.
Inobatanidzwa mukuona zvinovaka muviri, kuisa insulin signaling, uye maitiro ekugadzirisa metabolic.
Yakabatana nekushandiswa kwesimba, metabolism yemafuta, uye nzira dzekugadzirisa metabolism.
Kubatanidzwa kwekushanda kwema receptor system matatu aya kunoita kuti Retatrutide ive imwe yenzvimbo dzakasiyana dzekutsvagisa dzinoongorora mashandiro akaomarara emetabolism uye mhinduro dzemuviri dzinoenderana nemaitiro akawanda.
Retatrutide yave nyaya inokosha munzvimbo dzakasiyana-siyana dzekutsvaga kwesainzi, kusanganisira:
Vaongorori vanoramba vachiongorora chimiro chayo che "triple-agonist" chakasiyana uye zvazvinogona kuita pakukura kwepeptide mune ramangwana.
Boka rega rega reRetatrutide rinofanira kuongororwa zvakadzama, kusanganisira:
Chitupa Chekuongorora (COA) chinogona kupihwa kana chakumbirwa kuti chive nechokwadi chekuti chigadzirwa chacho chakanaka uye kuti chinoteverwa zvakanaka.
Kuti peptide irambe yakasimba zvakakwana:
Kuchengetedza Kwenguva Refu
Mushure meKugadziriswazve kweBumbiro reMitemo
Mamiriro ekuchengetedza akakodzera anobatsira kuchengetedza kuvimbika kwepeptide uye kushanda kwekuongorora.
Sarudzo dzekurongedza dziripo dzingasanganisira:
Huwandu hwakawanda uye mabasa eOEM ekurongedza anowanikwa kumasangano ane hunyanzvi hwekutsvagisa.
Retatrutide inopihwa chete pakutsvaga murabhoritari uye pakuongorora chete. Chigadzirwa ichi hachibvumidzwe kudyiwa nevanhu, kushandiswa mukurapa, kushandiswa pakurapa, kana nzira dzekuongorora. Vaongorori vane basa rekuona kuti mitemo yese inoshanda uye nhungamiro dzesangano dzinotevedzwa.